Our GPCR Assay Catalogue offers over 435 recombinant G protein coupled receptors (GPCR) expressed in stable cell lines and validated in over 840 binding and functional assays.
Characterization of your compounds in one or more of our assays (cAMP, IP-One, Aequorin, GTPgS, ERK1/2, Radioligand Binding assay, or customized assays) to determine agonist, antagonist or allosteric modulator potency, efficacy and functional selectivity with your data returned 5 days after compound delivery for repetitive testing.
Next to this extensive GPCR offer, we also provide ion channel or enzymatic assays, including kinases, as well as tailor-made assay development with a quick turnaround time. So if you do not find exactly what you are looking for, feel free to contact us and we'll work together to design the most fitting experiment with the most relevant target to address your research needs.
*: Receptors could have limited access due to patent restrictions in certain territories
**: this assay is performed using fluorescent calcium measurement
***: means that the cell line is available for functional assay. It has been validated for mRNA, cell surface expression and constitutive activity but not with a ligand
HS = Homo Sapiens ; MM = Mus Musculus ; RN = Rattus Norvegicus ; CF = Canis Familiaris ; CP = Guinea Pig (Cavia Porcellus) ; RH = Rhesus monkey (Macacca Mulatta) ; OC = Oryctolagus cuniculus